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VitabaseIngredientes

raíz de forskohlii

Condiciones de Salud27
Tabla de contenidos

Otros Nombres

Abyssinian coleusAlumãBalakahBlue spur flowerBoldo brasileiroBoldo gaúchoBoldo-da-terraBoldo-de-jardimBoldo-do-reinoBoldo-graúdoBoldo-peludoBoldo-veludoBrazilian boldoColeonolColeus adolfi-fridericiColeus barbatusColeus barbatus (Andrews) Benth. ex G.DonColeus coerulescensColeus forskalaeiColeus forskaleiColeus forskohliiColeus forskohlii (Willd.) Briq.Coleus penzigiiColeus speciosusColeus vestitusDolipraneFalse boldoFalso-boldoGandhe jharGandiraGarmarIndian coleusKarmeloKarpooravalliKarpuravalliMainmulMakandiMayinOcimum asperumOcimum hadienseOrthosiphon asperPanikoorkaPashan bhediPashanabhediPatharchurPlectranthus asperPlectranthus barbatusPlectranthus barbatus AndrewsPlectranthus coerulescensPlectranthus forskaoliiTapete-de-OxaláWoolly plectranthus

Sinopsis

Pau d'arco es un extracto herbal derivado de la corteza interna de varias especies de árboles sudamericanos, principalmente Tabebuia impetiginosa (también conocida como Handroanthus impetiginosus) y Tabebuia avellanedae. Ha sido valorado durante mucho tiempo en la medicina herbal tradicional por sus propiedades antimicrobianas, antiinflamatorias, estimulantes del sistema inmunitario y desintoxicantes. Los compuestos activos en el pau d'arco incluyen lapachol, beta-lapachona y quinoides, a los que se atribuyen los efectos biológicos de amplio espectro de la hierba.

Medicinalmente, el pau d'arco se utiliza como agente antimicrobiano natural, eficaz contra bacterias, virus, hongos (especialmente Candida albicans) y parásitos. A menudo se recomienda en la medicina integrativa para apoyar la desintoxicación, tratar infecciones crónicas por levaduras, reducir la inflamación sistémica y estimular la función inmunitaria.

También se utiliza para aliviar el dolor articular, los problemas gastrointestinales y las afecciones cutáneas como la psoriasis y el eccema. El pau d'arco está disponible en diversas formas, incluyendo té, cápsulas, tinturas y corteza en polvo. Es especialmente popular en los protocolos de limpieza y las dietas anticándida.

Algunos estudios sugieren un potencial antitumoral debido a la capacidad del lapachol para inhibir ciertas líneas de células cancerosas in vitro, aunque esta aplicación sigue siendo experimental y está limitada por preocupaciones sobre la toxicidad a dosis altas. Si bien generalmente es seguro en cantidades moderadas, el consumo excesivo puede causar náuseas, vómitos o adelgazamiento de la sangre, particularmente cuando se consume en forma de extractos concentrados.

Uso Histórico en Medicina
El pau d'arco tiene una larga historia de uso entre las tribus indígenas de la selva amazónica y las regiones andinas, como los pueblos inca, kallawaya y guaraní, quienes utilizaban la corteza interna para tratar infecciones, heridas, fiebres, problemas estomacales y mordeduras de serpiente. La corteza se decoccionaba frecuentemente como té o cataplasma y se aplicaba tópicamente o se consumía internamente.

Conocido como "taheebo" o "lapacho" en la medicina herbal tradicional sudamericana, el pau d'arco se utilizaba para tratar la malaria, la sífilis, la tuberculosis y las afecciones cutáneas inflamatorias. La madera en sí también era valorada por su resistencia y durabilidad, pero era la corteza interna la que los curanderos apreciaban por su potencial terapéutico.

El interés en el pau d'arco se extendió a Occidente en las décadas de 1960 y 1970, cuando los movimientos de salud natural comenzaron a explorar los botánicos amazónicos y andinos. Se volvió popular en los círculos herbales y naturopáticos como remedio natural para las infecciones crónicas, la debilidad inmunitaria y el apoyo a la desintoxicación. Durante ese tiempo, también fue promovido—aunque de manera controvertida—como una terapia complementaria contra el cáncer, debido a los estudios preliminares de laboratorio sobre el lapachol.

Condiciones de Salud

Condiciones de salud que raíz de forskohlii puede ayudar a apoyar.

  • Abuso y TraumaCientífico

    Forskolin raises intracellular cAMP, which inhibits mast cell degranulation and the release of histamine and allergic mediators such as leukotrienes. Preclinical (animal) studies show dose-dependent prevention of allergen-induced bronchospasm. This mechanism underlies long-standing traditional Ayurvedic use for allergic respiratory complaints and is supported by limited human asthma trials.

  • EdemaCientífico

    Forskohlii root (Coleus forskohlii) and its active diterpene forskolin activate adenylate cyclase to raise intracellular cAMP, relaxing bronchial smooth muscle. A single-blind RCT in 40 asthma patients found oral forskolin (10 mg/day for 6 months) reduced asthma attacks in 40% vs. 85% in the cromoglycate group. It has traditional use in Ayurvedic medicine for respiratory disorders.

  • HipoglucemiaCientífico

    Forskolin inhibits platelet aggregation in vitro via cAMP elevation in platelets, reducing thromboxane A2-mediated activation. Platelet aggregation inhibitory activity is listed as a confirmed pharmacological property in peer-reviewed literature.

  • HipotensiónCientífico

    Forskolin causes vasodilation by raising cAMP in vascular smooth muscle cells, lowering systemic vascular resistance. Small clinical studies from the 1980s–1990s demonstrated modest blood pressure reductions in humans, and the Godard 2005 RCT measured blood pressure as a secondary endpoint in overweight men.

  • Forskolin raises cAMP in pancreatic beta cells, enhancing glucose-stimulated insulin release and improving insulin sensitivity markers in human studies. A 12-week RCT in overweight/obese subjects showed significant improvement in insulin concentration and insulin resistance compared to placebo.

  • Forskolin activates adenylate cyclase similarly to parathyroid hormone signalling in bone cells, and a 12-week RCT in overweight men found a statistically significant increase in bone mass in the forskolin group versus placebo as measured by DXA. This represents the first in vivo human evidence for this effect.

  • AnginaCientífico

    Forskohlii root (Coleus forskohlii root) provides the diterpene forskolin and is cited in peer-reviewed dermatological literature and clinical studies as a validated anti-cellulite active, named as an ingredient with well-documented anti-cellulite activity in a published double-blind, placebo-controlled RCT and in MDPI Cosmetics 2026.

  • ApendicitisCientífico

    Forskolin demonstrates anti-inflammatory properties in laboratory and animal settings by raising cAMP, which broadly suppresses pro-inflammatory mediator release. Intraoperative infusion of a water-soluble forskolin derivative (colforsin daropate) showed anti-inflammatory effects in human cardiac surgery. Preclinical evidence is strong; dedicated anti-inflammatory RCTs in humans are lacking.

  • Intracavernosal injection of forskolin has been investigated as a treatment for vasculogenic erectile dysfunction, as cAMP promotes smooth muscle relaxation and penile blood flow. Small human studies suggest efficacy when administered by direct injection.

  • CulturismoCientífico

    Forskolin eye drops lower intraocular pressure by reducing aqueous humor production, providing neuroprotection to retinal ganglion cells. Multiple clinical trials, including a double-blind RCT in open-angle glaucoma patients, confirm IOP-reducing efficacy.

  • Forskolin eye drops reduce IOP by suppressing aqueous humor formation via cAMP elevation in ciliary epithelium. Multiple clinical trials including a double-blind RCT in 90 open-angle glaucoma patients confirm significant IOP reduction. Oral supplementation in combination formulas has also shown benefit.

  • Forskohlii root is the botanical source of forskolin and shares the same evidence base as Coleus forskohlii extract. Clinical trials show significant decreases in body fat and increases in lean body mass in obese men at 500 mg/day (10% extract) over 12 weeks. Traditional Ayurvedic medicine used the root for obesity and metabolic disorders.

  • JuanetesCientífico

    Forskolin is a positive inotrope that raises cAMP in cardiac muscle, increasing contractility. Two clinical trials using intravenous forskolin found positive cardiovascular effects in heart failure patients. A water-soluble derivative (colforsin daropate) is approved in Japan for acute heart failure.

  • Olor de piesCientífico

    A 12-week double-blind RCT found significant improvement in insulin concentration and insulin resistance in overweight/obese subjects receiving C. forskohlii extract. cAMP-mediated enhancement of beta-cell signalling and reduced adiposity are the proposed mechanisms.

  • Forskohlii root (from Coleus forskohlii) contains the bronchodilatory compound forskolin that raises bronchial smooth muscle cAMP, producing airway relaxation. Ayurvedic tradition and modern pharmacological data both support its use for asthma and respiratory conditions.

  • GingivitisCientífico

    A 12-week RCT specifically evaluated C. forskohlii extract in overweight/obese subjects for metabolic syndrome risk factors, finding improvements in insulin resistance and HDL-cholesterol. Reductions in body fat and blood pressure have been noted across multiple trials.

  • Forskolin increases cAMP-driven lipolysis via hormone-sensitive lipase activation, promotes thermogenesis, and may mildly stimulate thyroid hormone secretion. Multiple human RCTs show reductions in body fat percentage and fat mass, with one 12-week DBPC trial in men showing significant decreases versus placebo by DXA.

  • A 12-week double-blind RCT in overweight/obese men showed significantly increased serum free testosterone in the forskolin group versus placebo. cAMP elevation in Leydig cells is the proposed mechanism, as cAMP drives testosterone biosynthesis.

  • InfertilidadCientífico

    Forskohlii root (Coleus forskohlii root) is the botanical source of forskolin, the primary non-stimulant thermogenic compound that activates adenylyl cyclase to increase cAMP, triggering lipolysis and thermogenesis. Clinical trials show body composition improvements. Classified as a non-stimulant thermogenic in the 2016 Phytotherapy Research review.

  • Coleus forskohlii is documented across Ayurvedic, Siddha, and Unani traditions for chest pain (angina), attributed to its vasodilatory and antispasmodic pharmacology. No human RCTs specifically targeting angina have been published.

  • C. forskohlii is documented in Ayurvedic medicine for painful urination and bladder conditions. Forskolin's smooth muscle relaxant action on detrusor and urinary smooth muscle provides pharmacological plausibility, but no human clinical trials for bladder conditions exist.

  • EndometriosisTradicional

    C. forskohlii is historically documented in Ayurvedic medicine for bronchitis, sharing mechanistic overlap with its asthma indication via airway smooth-muscle relaxation. No clinical trials specifically for bronchitis have been identified.

  • Eczema is associated with reduced cAMP levels in skin and bronchial cells, leading to mast cell degranulation and inflammation. Forskolin's cAMP-raising mechanism is theoretically relevant and the plant has documented Ayurvedic use for eczema, but no direct human clinical trials for eczema have been conducted.

  • PulgasTradicional

    Forskolin's documented spasmolytic action on intestinal smooth muscle underlies its Ayurvedic use for intestinal colic and spastic conditions including IBS. The EBSCO Research Starters explicitly list IBS (spastic colon) among proposed uses. No human clinical trials for IBS have been published.

  • Forskolin's potent smooth-muscle relaxant (antispasmodic) action, mediated by cAMP elevation in uterine smooth muscle, underpins long-documented Ayurvedic use of C. forskohlii for dysmenorrhea. No human clinical trials have specifically evaluated the herb for menstrual cramps.

  • Psoriasis involves abnormally rapid skin cell proliferation linked to low cAMP and elevated cGMP. Forskolin's cAMP-raising mechanism is pharmacologically relevant, and C. forskohlii has long been used in Ayurveda for psoriasis. Experimental studies in mice support anti-psoriatic activity, but no human RCT has been conducted.

  • C. forskohlii is listed in Ayurvedic texts for urinary tract conditions including painful urination and urinary tract infections. Smooth muscle relaxation in the urinary tract is the proposed mechanism. No clinical trials for UTI or urinary tract health have been published.

Sistemas Corporales

Sistemas corporales que raíz de forskohlii puede ayudar a apoyar.

  • No hay sistemas corporales disponibles.
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